J. Lindman, A. Yadav, J. Gising, M. Larhed*: Two-chamber aminocarbonylation of aryl
bromides and triflates using amino acids as nucleophiles.
J. Org. Chem. 88 (2023), 12978-12985. DOI: 10.1021/acs.joc.3c00972
J. Wannberg, J. Gising, M. Henriksson, D. D. Vo, J. Sävmarker, J. Sallander, H. Gutiérrez-de Terán, J. Larsson, S. Hamid, H. Ablahad, I. Spizzo, T. A. Gaspari, R. E. Widdop, A. Grönbladh, N. N. Petersen, M. Backlund, M. Hallberg, M. Larhed*: N-(Heteroaryl)thiophene sulfonamides as angiotensin AT2 receptor ligands.
Eur. J. Med. Chem. 265 (2024) 116122 (11 p). DOI: 10.1016/j.ejmech.2024.116122
K. Engen, T. Lundbäck, A. Yadav, S. Puthiyaparambath, U. Rosenström, J. Gising, A. Jenmalm-Jensen, M. Hallberg, M. Larhed*: Inhibition of Insulin-regulated Aminopeptidase by Imidazo[1,5-α]pyridines; Synthesis and Evaluation.
Int. J. Mol. Sci. 25 (2024) 2516 (30 p). DOI: org/10.3390/ijms25052516
J. Beveridge, M. Söderström, R. Prieto-Díaz, H. Gutierrez-de-Teran, L. R. Odell, M. Hallberg, M. Larhed*, J. Gising*: Benzylhydroxamic Acids as Inhibitors of Insulin Regulated Aminopeptidase (IRAP).
Eur. J. Med. Chem. Rep. 12 (2024) 100215 (11 p). DOI: org/10.1016/j.ejmcr.2024.100215
J. Beveridge, M. Söderström, R. Prieto-Díaz, H. Gutierrez-de-Teran, L. R. Odell, M. Hallberg, M. Larhed*, J. Gising*: Benzylhydroxamic acids as IRAP Inhibitors: Sulfonamide Variations.
SynLett, 36 (2025) 2666-2670. DOI: org/10.1055/a-2562-7204
J. Lindman, S. Puthiyaparambath, J. Gising, L. R. Odell, M. Larhed*: A diastereoselective Mizoroki-Heck reaction for synthesis of spirooxindole-based unnatural amino acids using a Boc-protected amine as chiral auxiliary.
SynLett, 36 (2025) 2009-2013. DOI: 10.1055/a-2564-4920
J. Gising, J. Wannberg, R. Isaksson, J. Sallander, H. Gutiérrez-de-Terán, M. Backlund, M. Hallberg and M. Larhed*. New high affinity AT2 receptor ligands comprising a 2-methyl substituted phenylthiophene scaffold.
Bioorg. Med. Chem. 140 (2026) 118710 (6 p). DOI: 10.1016/j.bmc.2026.118710